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β-Nicotinamide Adenine Dinucleotide Phosphate Disodium Tote CAS: 24292-60-2
β-Nicotinamide Adenine Dinucleotide Phosphate Disodium ToteHe coenzyme e horapa whānuitia ana i roto i ngā mea ora, e whai wāhi ana ki ngā tauhohenga waikura-whakaiti. He kaikawe irahiko ia i roto i ngā tauhohenga maha, ka waikurahia (NADP+) me te whakaitihia (NADPH).β-Nicotinamide Adenine Dinucleotide Phosphate Disodium ToteHe matū tēnei e herea ana te waikawa nicotinic, te amide adenine dinucleotide, me te ngota phosphate mā te here ester. He kaiwhakawhiwhi hauwai, ā, ka taea te whakamahi mō te whakawhanake me te whakawhanake i ngā momo matū tātaritanga in vitro.
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β-Nicotinamide Adenine Dinucleotide Lithium tote (NAD Lithium tote) CAS:64417-72-7
β-Nicotinamide Adenine Dinucleotide tote lithiumHe coenzyme matua ki te pākia o te tinana. Kei roto i ngā pūtau ora katoa, ka kiia te NAD he dinucleotide nā te mea e rua ngā nucleotide e honoa ana mā roto i ō rātou rōpū phosphate. Kei roto i tētahi nucleotide he adenine nucleobase, ā, kei roto i tētahi he nicotinamide. E rua ngā āhua o te NAD: he āhua kua waikuratia, he āhua kua whakaititia, e whakarapopototia ana ko NAD+ me NADH (H mō te hauwai).
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Venlafaxine CAS:93413-69-5
He rongoā ārai pouri te Venlafaxine nō te akomanga serotonin me te norepinephrine reuptake inhibitor (SNRI). I whakawhanakehia tuatahitia tēnei rongoā e Wyeth i te 19Chemicalbook93, ā, kei te hokohokohia inaianei e Pfizer. Kua whakaaetia tēnei rongoā mō te rongoā i te mate pouri nui (MDD), te mate manukanuka whānui (GAD), me te pouri e pā ana ki te manukanuka.
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Ciclopirox Ethanolamine CAS:41621-49-2 Kaihanga Kaiwhakarato
He rongoā anti-harore whānui te Ciclopirox ethanolamine, ā, he kaha patu huakita anō hoki tōna ki te maha o ngā huakita Gram-pai me Gram-kino, ā, he āhuatanga ārai-mumura anō hoki. E whakamahia ana hei rongoā ā-papa mō ngā mate kiri harore me ngā mate whao.
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Desvenlafaxine Succinate CAS:386750-22-7
Ko te Desvenlafaxine Succinate he aukati rua mō te serotonin me te norepinephrine reuptake (SNRI) i whakaaetia mō te rongoā i te mate pouri nui (MDD) i te United States i te tau 2008. Hei whakapai ake i te whai huatanga me te haumaru o te venlafaxine, i kitea e Wyeth, ā, i whakawhanakehia hoki e ia tētahi o ngā matū nui o te venlafaxine, arā, ko te matū O-desmethyl (desvenlafaxine).
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Doxazosin Mesylate CAS:77883-43-3 Kaihanga Kaiwhakarato
Ko te Doxazosin mesylate he matū quinazoline he aukati whiriwhiri i te momo alpha1 o ngā kaiwhakawhiwhi alpha adrenergic. Ko te Doxazosin mesylate he whakatupuranga hou o te aukati kaiwhakawhiwhi quinazolone α1 i whakawhanakehia e te kamupene Pfizer (Te Hononga o Amerika). He roa te haurua-ora, e whakaatu ana i ōna pānga ki te whakawhānui i ngā oko toto, te whakaiti i te ātete o ngā oko toto me te whakaheke i te toto toto mā te aukati i te kaiwhakawhiwhi a1. Kua tūtohutia ki tāwāhi hei rongoā haumanu tuatahi mō te whakaheke toto toto tiketike me te maimoatanga o te mate prostate.
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L-Isoleucine CAS:73-32-5 Kaihanga Kaiwhakarato
Ko te L-Isoleucine, e mōhiotia ana ko te Isoleucine, he waikawa amino he isomer o te leucine. He mea nui ki te hanga hemoglobin me te whakahaere i te huka toto me ngā taumata pūngao. Ko te L-Isoleucine he isomer o te L-leucine, ā, he waikawa amino nui. Ka hangaia mai i te threonine, ā, he waikawa amino mekameka peka-waikura.
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Captopril CAS:62571-86-2 Kaihanga Kaiwhakarato
Ko Captopril te mea tino rangahautia o ngā aukati whākōkī-hurihuri angiotensin kua whakaarohia hei rongoā whakaheke toto. Ka aukati i te whākōkī-hurihuri angiotensin, e pehi ana i te hanganga o te angiotensin II, ā, ka whakamama i tōna pānga whakaheke toto ki ngā oko toto me ngā oko toto. Ka whakaitihia te taumahatanga ā-taha o ngā oko toto, ā, ka heke te pēhanga toto.
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Candesartan CAS:139481-59-7 Kaihanga Kaiwhakarato
He kaitukino angiotensin II receptor I (AT1) a Candesartan, IC50s=1.12 me te 2.86 nM mō te cortex adrenal kau me te aorta rāpeti. Ka ārai i te whakahekenga o ngā rīpene aorta rāpeti nā te angiotensin II, kāore he pānga ki te whakahekenga i puta mai i ētahi atu kaihoko pērā i te norepinephrine, KCl, serotonin, PGF2α, endothelin rānei.
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Candesartana Cilexetila CAS:145040-37-5
Ko te Candesartan Celexetil he rite ki te ester o te angiotensin II antagonist Candesartan (sc-217825). Mā te ārai i tēnei kaiwhakawhiwhi ka ārai i te here o te angiotensin II, he mea whakapūmau i te toto. Ko te pānga whānui o tēnei ko te whakanui i te toto me te whakanui ake i te rōrahi toto capillary. Ko te Candesartan Celexetil Ester he aukati i te AT1.
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Bupropion CAS:34911-55-2 Kaihanga Kaiwhakarato
He ketone kakara te Bupropion, he propiophenone e mau ana i te rōpū tert-butylamino i te tūranga 2 me te chloro substituent i te tūranga 3 i runga i te mowhiti phenyl. He mahi tōna hei rongoā ārai pouri, hei poke taiao, hei xenobiotic hoki. He matū amino tuarua, he mema nō ngā monochlorobenzenes me te ketone kakara.
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Bezafibrate CAS:41859-67-0 Kaihanga Kaiwhakarato
Ko te Bezafibrate he amide waikawa monocarboxylic i whiwhihia mā te whakakotahitanga ōkawa o te rōpū carboxy o te waikawa 4-chlorobenzoic me te rōpū amino o te waikawa 2-[4-(2-aminoethyl)phenoxy]-2-methylpropanoic. Ka whakamahia te Benafibrate hei rongoā mō te hyperlipidemia. He mahi āna hei xenobiotic, hei poke taiao, hei geroprotector me hei rongoā antilipemic. He waikawa monocarboxylic, he ether kakara, he mema o ngā monochlorobenzenes me te amide waikawa monocarboxylic. He hononga mahi tōna ki te waikawa propionic.
