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Tetracycline CAS:60-54-8
He paturopi whānui te Tetracycline nō te akomanga tetracycline, i ahu mai i te matū tūturu chlortetracycline. Ka aukati i te hanganga pūmua huakita mā te herea ki te ribosome huakita, ā, ka ārai i te piri o te aminoacyl-tRNA ki te matatini mRNA-ribosome. Mā tēnei tikanga mahi ka hua ake he pānga bacteriostatic ki te whānuitanga o ngā huakita gram-pai me ngā huakita gram-kino, tae atu ki ētahi protozoa.
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Teicoplanin CAS:61036-62-2
Ko te Teicoplanin he paturopi glycopeptide i ahu mai i te Actinoplanes teichomyceticus, he whai hua ki ngā momo huakita karamu-pai tae atu ki te Staphylococcus aureus ātete-methicillin (MRSA). Ka aukati i te hanganga o te pakitara pūtau huakita mā te herea ki te pito D-alanyl-D-alanine o ngā matū peptidoglycan, ka hua ake te pakaru o te pūtau me ngā pānga patu huakita. He maha ngā wā ka whakamahia te Teicoplanin i roto i ngā tautuhinga haumanu hei rongoā i ngā mate kino i puta mai i ngā rauropi karamu-pai.
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Sulfisoxazol (4-amino-N-(3,4-dimethyl-5-isoxazolyl)benzenesulfonamide) CAS:127-69-5
Ko te Sulfisoxazole, e mōhiotia ana ko te sulfafurazole, he paturopi sulfonamide nō te akomanga rongoā sulfa. E whakaahuatia ana ko te 4-amino-N-(3,4-dimethyl-5-isoxazolyl)benzenesulfonamide, ka aukati te sulfisoxazole i te tipu o te huakita mā te whakararuraru i te hanganga o te waikawa folic. Ko tēnei tikanga mahi e aro ana ki te dihydropteroate synthase, he whākōkī e tika ana mō te hanga folate huakita, ā, ka aukati i tō rātou tipu me te horapa.
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Sulfapyridine CAS:144-83-2
Ko te Sulfapyridine he paturopi sulfonamide i whakamahia i mua hei rongoā i ngā mate kitakita, inā koa i te Pakanga Tuarua o te Ao. Nō roto i te akomanga o ngā rongoā sulfa, e aukati ana i te tipu o ngā kitakita mā te whakararuraru i te hanga o te waikawa folic. Ka puta ngā pānga bacteriostatic o te Sulfapyridine mā te aro ki te dihydropteroate synthase, he whākōkī nui mō te hanga folate i roto i ngā kitakita.
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Tazobactam CAS:89786-04-9
He aukati beta-lactamase a Tazobactam e whakarei ake ana i te mahi a ngā paturopi beta-lactam mā te tiaki i a rātou mai i te pirau e ngā whākōkī beta-lactamase i hangaia e te maha o ngā huakita ātete. He mea whakamahi noa i te taha o ngā paturopi beta-lactam pēnei i te piperacillin hei whakawhānui ake i tō rātou whānuitanga mahi ki ngā momo mate huakita. Ka whai hua a Tazobactam ki te whakahoki mai i te whai huatanga o ngā paturopi beta-lactam ki ngā huakita whakaputa beta-lactamase, inā koa ngā rauropi gram-negative.
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Tigecycline CAS:220620-09-7
Ko te Tigecycline he paturopi glycylcycline whānui-whānui e aukati ana i te hanganga pūmua huakita mā te herea ki te waeine ribosomal 30S, ā, ka puta he pānga bacteriostatic ki te whānuitanga o ngā huakita gram-pai me te gram-kino, tae atu ki ngā pathogens ātete-maha-rongoā. He whanaunga hanganga ki ngā tetracycline engari he kaha ake te mahi ki ngā momo ātete nā tōna tikanga mahi ahurei me ngā whakarerekētanga hanganga.
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Tote konutai Sulbactam CAS:69388-84-7
Ko te tote konutai Sulbactam he aukati beta-lactamase e whakamahia whānuitia ana me ētahi paturopi hei whawhai i ngā mate huakita. Mā te aukati i te mahi a ngā whākōkī beta-lactamase i hangaia e ngā huakita, ka kore ai e whai hua ngā paturopi. Mā te aukati i te pakaru o ngā paturopi pērā i ngā penicillin me ngā cephalosporin, ka āwhina te tote konutai sulbactam ki te whakarei ake i ō rātou āhuatanga patu huakita. He maha ngā wā ka whakamahia tēnei matū me ngā paturopi pērā i te ampicillin hei hanga i ngā pānga tahi ki te whānuitanga o ngā momo huakita ngoikore.
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Sulfadimidine CAS:57-68-1
Ko te Sulfadimidine, e mōhiotia ana ko te sulfamethazine, he paturopi sulfonamide e whakamahia ana hei rongoā i ngā mate kitakita. Nō te akomanga o ngā paturopi e mōhiotia ana ko ngā rongoā sulfa, e mahi ana mā te aukati i te tipu me te whakaputa uri o ngā kitakita. Ka whakararu te Sulfadimidine i te hanganga o te waikawa folic i roto i ngā kitakita, he wāhanga nui mō tō rātou oranga, ka hua ake he pānga bacteriostatic ki te whānuitanga o ngā kitakita gram-pai me ngā kitakita gram-kino.
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Tote konutai sulfacetamide CAS: 6209-17-2
Ko te tote konutai Sulfacetamide he matū wairewa-wai o te sulfacetamide, he paturopi sulfonamide e whakamahia whānuitia ana i roto i ngā whakatakotoranga kiri hei rongoā i ngā mate kitakita o te kiri me ngā kanohi. Ka whakarei ake tēnei momo tote i te wairewa me te pumau o te sulfacetamide, kia pai ai mō ngā tono rongoā. Ka mahi te tote konutai Sulfacetamide mā te aukati i te tipu o ngā kitakita, inā koa ko ērā e pāngia ana e ngā āhuatanga pēnei i te acne vulgaris, te seborrheic dermatitis, me ngā mate kanohi pēnei i te conjunctivitis. Ka whakararuraru i te hanganga folate kitakita, ka whai hua ki te whānuitanga o ngā kitakita gram-pai me te gram-kino.
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Streptomycin sulfate CAS: 3810-74-0
He rongoā paturopi te Streptomycin sulfate nō te akomanga aminoglycoside. I ahu mai i te huakita Streptomyces griseus, ā, e whakamahia whānuitia ana hei rongoā i ngā mate kitakita. Ka aukati te mahi a te Streptomycin sulfate i te hanganga pūmua kitakita, ā, ka patu pai i ngā kitakita ngoikore. He maha ngā wā ka tohua hei rongoā mō te mate kohi, te mate urutā, te tularemia, me ētahi atu mate i puta mai i ngā kitakita ngoikore. Ko te Streptomycin sulfate e wātea ana i roto i te ahua werohanga, ā, ka tukuna mā roto i te uaua, mā roto rānei i te uaua i raro i te tirotiro a te rata.
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Tote konutai sulfamethoxazole CAS: 4563-84-2
Ko te tote konutai Sulfamethoxazole he matū wairewa-wai o te sulfamethoxazole, he paturopi sulfonamide e whakamahia ana hei rongoā i ngā mate kitakita. Ka whakarei ake tēnei momo tote i te wairewa me te pumau o te sulfamethoxazole, kia pai ai mō ngā momo rongoā. Ka puta te pānga bacteriostatic o te tote konutai Sulfamethoxazole mā te aukati i te hanga o te waikawa folic i roto i ngā kitakita, he tukanga nui mō tō rātou tipu me te whakaputa uri. He whai hua ki te whānuitanga o ngā kitakita karamu-pai me ngā kitakita karamu-kino.
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Sulfamethoxazole CAS:723-46-6
Ko te Sulfamethoxazole he paturopi sulfonamide e whakamahia whānuitia ana me te trimethoprim hei hanga i tētahi rongoā paturopi kaha e mōhiotia ana ko te co-trimoxazole, trimethoprim-sulfamethoxazole rānei (TMP-SMX). Nō roto i te akomanga o ngā paturopi e mōhiotia ana ko ngā rongoā sulfa, e aukati ana i te tipu o ngā huakita mā te whakararuraru i te hanganga o te waikawa folic. Ka aro nui te Sulfamethoxazole ki te dihydropteroate synthase, he whākōkī e uru ana ki te hanga folate, ā, ka puta he pānga bacteriostatic ki te whānuitanga o ngā huakita gram-pai me ngā huakita gram-kino.
