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tert-butyl 4-hydroxy-3,4-dihydroquinoline-1(2H)-carboxylate CAS: 932398-74-8
Ko te Tert-butyl 4-hydroxy-3,4-dihydroquinoline-1(2H)-carboxylate, e mōhiotia whānuitia ana ko te pūhui Y, he pūhui matū maha-whakamahinga me ngā tono nui i roto i ngā ahumahi rongoā me te pūtaiao rauemi. Me te tauira ngota o C15H21NO3, kei roto i tēnei pūhui he tūāpapa quinoline ahurei kua whakakapia ki te rōpū tert-butyl me te mahi carboxylate. Ko tōna hanganga motuhake e whakarato ana i ngā āhuatanga e hiahiatia ana he mea nui mō ngā tono kanorau, mai i te hanganga rongoā ki te matū rauemi. Hei takawaenga matua i roto i te hanganga rauropi, he turanga mō te whanaketanga o ngā rongoā hou me ngā rauemi mahi, e akiaki ana i te auahatanga i roto i ngā momo rāngai.
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Semaglutide CAS:910463-68-2
He kaha te Semaglutide hei kaiwhakawhiwhi i te glucagon-like peptide-1 (GLP-1) e whakamahia ana hei rongoā i te mate huka momo 2 me te momona. He rite te hanganga ki te homoni GLP-1 taketake, ka roa te mahi rongoā a te semaglutide nā te mea kua whakarerekētia ki te mekameka taha waikawa ngako. Mā tōna tauira ngota C187H291N45O59, ka roa te haurua-ora o te semaglutide ka taea te horopeta kotahi i te wiki, ka pai ake te ngāwari o te tūroro me te piri ki ngā tikanga rongoā.
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Linaclotide CAS:851199-59-2
He agonist guanylate cyclase-C (GC-C) te Linaclotide e whakamahia ana mō te rongoā i te mate puku mārō me te mate puku irritable me te mate puku mārō (IBS-C). He rite te hanganga ki te peptide guanylin taketake, ka herea e te linaclotide ngā kaiwhakawhiwhi GC-C i roto i te ara gastrointestinal, ka whakahohehia hoki, ka hua ake te nui haere o te wai o te puku me te tere haere o te wā. Me tōna tauira ngota C59H79N15O21S6, ka tukuna e te linaclotide he huarahi whai kiko hei whakaora i te mate puku mārō me te whakamamae i te mamae o te puku e pā ana ki te IBS-C, hei whakapai ake i te kounga o te oranga o ngā tūroro.
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Liraglutide CAS:204656-20-2
He kaha te kaha o te Liraglutide hei kaiwhakawhiwhi i te glucagon-like peptide-1 (GLP-1) e whakamahia ana hei rongoā i te mate huka momo 2 me te momona. He rite te hanganga ki te homoni GLP-1 taketake, ka roa te mahi rongoā a te liraglutide nā te mea ka whakarerekētia ki te mekameka taha waikawa ngako. Mā tōna tauira ngota C172H265N43O51, ka roa te haurua-ora o te liraglutide ka taea te horopeta kotahi i te rā, ka pai ake te ngāwari o te tūroro me te piri ki ngā tikanga rongoā.
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etil 4-(hydroxymethyl)-1H-pyrazole-5-carboxylate CAS:61453-49-4
Ko te Ethyl 4-(hydroxymethyl)-1H-pyrazole-5-carboxylate, he matū maha-whakamahinga, he mea nui puta noa i ngā rāngai rongoā me ngā matū ahuwhenua. Me te tātai ngota C8H10N2O3, kei roto he mowhiti pyrazole kua whakakapia ki te rōpū ethyl, he wāhanga hydroxymethyl, me te mahi carboxylate. He takawaenga nui tēnei matū i roto i te hanganga rauropi, e āwhina ana i te whanaketanga o ngā momo rongoā me ngā matū ahuwhenua. Nā tōna hanganga ahurei me ngā rōpū mahi ka waiho hei poraka hanga maha-whakamahinga mō te hanga i ngā ngota me ngā tono rerekē, e akiaki ana i te auahatanga i roto i ngā ahumahi maha.
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Ethyl 4-cyanopiperidine-4-carboxylatehydrochloride CAS: 123730-64-3
Ko te Ethyl 4-cyanopiperidine-4-carboxylate hydrochloride, he matū nui, he mea nui i roto i ngā ahumahi rongoā me te ahuwhenua. Me te tātai ngota C9H14ClNO2, kei roto he mowhiti piperidine kua whakakapia ki te rōpū ethyl me te wāhanga cyano, me te mahi carboxylate, e herea katoa ana ki te ion chloride. He takawaenga nui tēnei matū i roto i te hanganga rauropi, e āwhina ana i te whanaketanga o ngā momo rongoā me ngā matū ahuwhenua. Nā tōna hanganga ahurei me ngā rōpū mahi ka waiho hei poraka hanga maha mō te hanga i ngā ngota me ngā tono rerekē, e whakatairanga ana i te auahatanga i roto i ngā rāngai maha.
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methyl imidazo[1,5-a]pyridine-7-carboxylate CAS:1377829-50-9
Ko te Methyl imidazo[1,5-a]pyridine-7-carboxylate, he matū kei roto te tātai ngota C9H7N3O2, e mōhiotia whānuitia ana mō ōna whakamahinga maha i roto i ngā mara rongoā me te pūtaiao rauemi. Kei roto i te anga imidazo-pyridine, e whakaatu ana i ngā āhuatanga hanganga ahurei e whai wāhi ana ki ōna whakamahinga kanorau. He takawaenga nui tēnei matū i roto i te hanganga rauropi, e mahi ana hei turanga mō te whanaketanga o ngā rongoā me ngā rauemi mahi. Nā tōna hanganga motuhake me tōna kaha tauhohenga e waiho ai hei wāhanga nui i roto i ngā mahi rangahau me ngā mahi ahumahi, e akiaki ana i te auahatanga puta noa i ngā rāngai rerekē.
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Arg34GLP-1 CAS:1169630-82-3
Ko te Arg34GLP-1, e mōhiotia ana ko te Arginine-34 Glucagon-Like Peptide 1, he homoni peptide bioactive e whai pānga nui ana ki te whakahaere i te pākia o te tinana me ngā wawaotanga rongoā mō te mate huka me te momona. I ahu mai tēnei peptide i te homoni glucagon-like peptide 1 (GLP-1) ā, kei roto he toenga arginine i te tūranga 34. Nā tōna hanganga ngota me ngā mahi koiora e pai ai te whakamahi mō ngā tono rongoā e aro ana ki te whakapai ake i te homeostasis glucose me te whakatairanga i te whakaheke taumaha.
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1-tert-Butyl 4-ethyl 4-cyanopiperidine-1,4-dicarboxylate CAS:1016258-66-4
Ko te 1-tert-Butyl 4-ethyl 4-cyanopiperidine-1,4-dicarboxylate he matū e mōhiotia ana mō ōna whakamahinga maha i roto i ngā ahumahi rongoā me te ahuwhenua. Me te tātai ngota C15H24N2O4, e whakaatu ana i tētahi whakaritenga hanganga ahurei e whakaatu ana i tētahi mowhiti piperidine kua whakakapia ki ngā rōpū tert-butyl, ethyl, me te cyano. He takawaenga nui tēnei matū i roto i te hanganga rauropi, e whai wāhi nui ana ki te whanaketanga o ngā rongoā me ngā matū ahuwhenua kanorau. Nā tōna tauira whakakapinga rautaki me ngā rōpū mahi ka waiho hei poraka hanga maha mō te hanga i ngā hanganga ngota matatini me ngā āhuatanga e hiahiatia ana mō ngā tono rerekē.
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6-Kōro-3,4-dihydro-2H-benzo[b][1,4]oxazine hydrochloride CAS:1956310-17-0
Ko te 6-Chloro-3,4-dihydro-2H-benzo[b][1,4]oxazine hydrochloride, e mōhiotia whānuitia ana ko te pūhui X, he pūhui matū e maha ana ngā whakamahinga i roto i ngā ahumahi rongoā me te pūtaiao rauemi. Me te tauira ngota o C8H8ClNO•HCl, kei roto i tēnei pūhui he tūāpapa benzo[b][1,4]oxazine ahurei kua whakakapia ki te ngota chlorine. Nā tōna hanganga motuhake ka waiho hei takawaenga whai hua i roto i te hanganga rauropi, hei turanga mō te whanaketanga o ngā momo rongoā me ngā rauemi mahi.
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8-Methylquinazolin-4(3H)-one CAS:19181-54-5
He matū te 8-Methylquinazolin-4(3H)-one, he maha ngā whakamahinga i roto i te matū rongoā me te rangahau rongoā. Nā tōna tauira ngota C9H8N2O, nō te akomanga quinazolinone o ngā matū, ā, he āhuatanga ā-tinana, ā-matū ahurei e whai hua ai mō ngā mahi kimi rongoā me ngā rangahau whanaungatanga hanganga-mahi i roto i te whanaketanga o ngā kaihoko rongoā hou.
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5,6-Difluoro-2,3-dihydro-1H-isoindol-1-one CAS:1192040-50-8
Ko te 5,6-Difluoro-2,3-dihydro-1H-isoindol-1-one, e mōhiotia ana mō ōna āhuatanga maha-whakamahinga, he matū nui i roto i ngā mahi rangahau me ngā mahi ahumahi. Mā te tauira matū C8H6F2NO, kei roto he matua isoindolone ahurei kua whakakapia ki ngā ngota fluorine e rua, e whakarato ana i ngā āhuatanga motuhake ki tōna hanganga. Ka kitea ngā tono o tēnei matū puta noa i ngā mara rerekē nā tōna kaha ki te tauhohe me te kaha ki te hanga i ngā ngota matatini e pā ana ki te rongoā me te pūtaiao rauemi.
